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Tracazolate hydrochloride

CAS No. 1135210-68-2

Tracazolate hydrochloride ( Tracazolate (hydrochloride) )

产品货号. M27728 CAS No. 1135210-68-2

Tracazolate hydrochloride is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity.

纯度: >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
规格 价格/人民币 库存 数量
2MG ¥292 有现货
5MG ¥478 有现货
10MG ¥778 有现货
25MG ¥1596 有现货
50MG ¥2657 有现货
100MG ¥3993 有现货
200MG 获取报价 有现货
500MG 获取报价 有现货
1G 获取报价 有现货

生物学信息

  • 产品名称
    Tracazolate hydrochloride
  • 注意事项
    本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
  • 产品简述
    Tracazolate hydrochloride is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity.
  • 产品描述
    Tracazolate hydrochloride is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity. Tracazolate hydrochloride potentiates α1β1γ2s and α1β3γ2 with EC50s of 13.2 μM and 1.5 μM.(In Vitro):Tracazolate hydrochloride (10 μM) enhanced the sensitivity of α1β2δ-containing GABAA receptors and increased the maximum current amplitude in oocytes . Tracazolate hydrochloride inhibited α1β1ε, α1β3ε, α1β3, and α6β3γ with EC50s of 4.0 μM, 1.2 μM, 2.7 μM, and 1.1 μM. Tracazolate hydrochloride interacted with γ-aminobutyric acid GABAA receptors, adenosine receptors, and phosphodiesterases .
  • 同义词
    Tracazolate (hydrochloride)
  • 通路
    Others
  • 靶点
    Other Targets
  • 受体
    ——
  • 研究领域
    ——
  • 适应症
    ——

化学信息

  • CAS Number
    1135210-68-2
  • 分子量
    340.9
  • 分子式
    C16H25ClN4O2
  • 纯度
    >98% (HPLC)
  • 溶解度
    ——
  • SMILES
    Cl.CCCCNc1c(C(=O)OCC)c(C)nc2n(CC)ncc12
  • 化学全称
    ——

运输与储存

  • 储存条件
    (-20℃)
  • 运输条件
    With Ice Pack
  • 稳定性
    ≥ 2 years

参考文献

1.King HL Jr, Dyar RE, Wilken DR. Ketopantoyl lactone and ketopantoic acid reductases. Characterization of the reactions and purification of two forms of ketopantoyl lactone reductase. J Biol Chem. 1974 Aug 10;249(15):4689-95.
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